ChemSpider 2D Image | Fentanyl citrate | C28H36N2O8

Fentanyl citrate

  • Molecular FormulaC28H36N2O8
  • Average mass528.594 Da
  • Monoisotopic mass528.247192 Da
  • ChemSpider ID13213

More details:






Validated by Experts, Validated by Users, Non-Validated, Removed by Users

213-588-0 [EINECS]
2-Hydroxy-1,2,3-propantricarbonsäure --N-phenyl-N-[1-(2-phenylethyl)-4-piperidinyl]propanamid (1:1) [German] [ACD/IUPAC Name]
2-Hydroxypropan-1,2,3-tricarbonsäure--N-phenyl-N-[1-(2-phenylethyl)piperidin-4-yl]propanamid(1:1)
990-73-8 [RN]
Acide 2-hydroxy-1,2,3-propanetricarboxylique - N-phényl-N-[1-(2-phényléthyl)-4-pipéridinyl]propanamide (1:1) [French] [ACD/IUPAC Name]
acide 2-hydroxypropane-1,2,3-tricarboxylique - N-phényl-N-[1-(2-phényléthyl)pipéridin-4-yl]propanamide (1:1)
ACTIQ [Trade name]
FENTANEST [Trade name]
Fentanyl citrate [JAN] [JP15] [USAN] [USP]
Leptanal
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Validated by Experts, Validated by Users, Non-Validated, Removed by Users

D01399 [DBID]
DEA No. 9801 [DBID]
R 5240 [DBID]
UN2810 [DBID]
  • Experimental Physico-chemical Properties
  • Miscellaneous
    • Chemical Class:

      The citric acid salt of fentanyl, comprising equimolar amounts of citric acid and fentanyl. A <greek>mu</greek>-opioid receptor agonist, it is a potent opioid analgesic used in the management of labou r pain, postoperative pain, and chronic intractable cancer pain. It is also widely used as the analgesic component of balanced anaesthesia. ChEBI CHEBI:31602
    • Bio Activity:

      7-TM Receptors Tocris Bioscience 3247
      Mu Opioid Receptors Tocris Bioscience 3247
      Opioid Receptors Tocris Bioscience 3247
      Potent and selective ? agonist Tocris Bioscience 3247
      Potent and selective ?-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for ?-, ?- and ?-opioid receptors respectively). Displays antinociceptive activity in vivo. Tocris Bioscience 3247
      Potent and selective mu agonist Tocris Bioscience 3247
      Potent and selective mu-opioid receptor agonist (Ki values are 7.0, 151 and 470 nM for mu-, delta- and kappa-opioid receptors respectively). Displays antinociceptive activity in vivo. Tocris Bioscience 3247

Predicted data is generated using the ACD/Labs Percepta Platform - PhysChem Module

No predicted properties have been calculated for this compound.

Click to predict properties on the Chemicalize site





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