ChemSpider 2D Image | Rivoceranib Mesylate | C25H27N5O4S

Rivoceranib Mesylate

  • Molecular FormulaC25H27N5O4S
  • Average mass493.578 Da
  • Monoisotopic mass493.178375 Da
  • ChemSpider ID28294976

More details:






Validated by Experts, Validated by Users, Non-Validated, Removed by Users

Acide méthanesulfonique - N-[4-(1-cyanocyclopentyl)phényl]-2-[(4-pyridinylméthyl)amino]nicotinamide (1:1) [French] [ACD/IUPAC Name]
Methansulfonsäure --N-[4-(1-cyancyclopentyl)phenyl]-2-[(4-pyridinylmethyl)amino]nicotinamid (1:1) [German] [ACD/IUPAC Name]
Rivoceranib Mesylate
1218779-75-9 [RN]
3-Pyridinecarboxamide, N-[4-(1-cyanocyclopentyl)phenyl]-2-[(4-pyridinylmethyl)amino]-, methanesulfonate (1:1) [ACD/Index Name]
811803-05-1 [RN]
Apatinib [Wiki]
Apatinib (YN968D1)
Apatinib Mesylate
apatinib mesylate
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Validated by Experts, Validated by Users, Non-Validated, Removed by Users

TK02X14ASJ [DBID]
UNII:TK02X14ASJ [DBID]
UNII-TK02X14ASJ [DBID]
  • Experimental Physico-chemical Properties
  • Miscellaneous
    • Target Organs:

      VEGFR inhibitor TargetMol T2582
    • Bio Activity:

      Apatinib(YN-968D1) is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM. MedChem Express
      Apatinib(YN-968D1) is an orally bioavailable, selective VEGFR2 inhibitor with IC50 of 1 nM.;IC50 value: 1 nM;Target: VEGFR2Apatinib, also known as YN968D1, is a tyrosine kinase inhibitor that selectively inhibits the vascular endothelial growth factor receptor-2 (VEGFR2, also known as KDR). It is an orally bioavailable, small molecule agent which is thought to inhibit angiogenesis in cancer cells; specifically apatinib inhibits VEGF-mediated endothelial cell migration and proliferation thus blocking new blood vessel formation in tumor tissue. This agent also mildly inhibits c-Kit and c-SRC tyrosine kinases. MedChem Express HY-13342
      Protein Tyrosine Kinase/RTK; MedChem Express HY-13342
      Tyrosine Kinase/Adaptors TargetMol T2582
      VEGFR MedChem Express HY-13342
      VEGFR2;Ret;c-kit;c-Src; TargetMol T2582

Predicted data is generated using the ACD/Labs Percepta Platform - PhysChem Module

No predicted properties have been calculated for this compound.

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