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- Opioid ligands with mixed properties from substituted enantiomeric N-phenethyl-5-phenylmorphans. Synthesis of a µ-agonist δ-antagonist and δ-inverse agonists. Kejun Cheng, In Jong Kim, Mei-Jing Lee, Steven A. Adah, Tyler J. Raymond, Edward J. Bilsky, Mario D. Aceto, Everette L. May, Louis S. Harris, Andrew Coop, Christina M. Dersch, Richard B. Rothman, Arthur E. Jacobson, Kenner C. Rice
, Org. Biomol. Chem.
, 2007
, 5
, 1177
- Comprehensive overview of biased pharmacology at the opioid receptors: biased ligands and bias factors. Jolien De Neve, Thomas M. A. Barlow, Dirk Tourwé, Frédéric Bihel, Frédéric Simonin, Steven Ballet
, RSC Med. Chem.
, 2021
, 12
, 828
- A homogeneous single-label quenching resonance energy transfer assay for a δ-opioid receptor–ligand using intact cells. Kari Kopra, Shweta, Eija Martikkala, Pekka Hänninen, Ulla Petäjä-Repo, Harri Härmä
, Analyst
, 2013
, 138
, 4907
- Synthesis and pharmacological evaluation of enantiomerically pure endo-configured KOR agonists with 2-azabicyclo[3.2.1]octane scaffold. Hendrik Jonas, Daniele Aiello, Bastian Frehland, Kirstin Lehmkuhl, Dirk Schepmann, Jens Köhler, Patrizia Diana, Bernhard Wünsch
, Org. Biomol. Chem.
, 2021
, 19
, 8384
- Effects of polar κ receptor agonists designed for the periphery on ATP-induced Ca2+ release from keratinocytes. Fabian Galla, Christian Bourgeois, Kirstin Lehmkuhl, Dirk Schepmann, Michael Soeberdt, Tobias Lotts, Christoph Abels, Sonja Ständer, Bernhard Wünsch
, Med. Chem. Commun.
, 2016
, 7
, 317
- Synthesis of diarylmethylamines via palladium-catalyzed regioselective arylation of 1,1,3-triaryl-2-azaallyl anions. Minyan Li, Baris Yücel, Javier Adrio, Ana Bellomo, Patrick J. Walsh
, Chem. Sci.
, 2014
, 5
, 2383
- Diastereoselective synthesis of conformationally restricted KOR agonists. Denise Ilari, Sarah Maskri, Dirk Schepmann, Jens Köhler, Constantin G. Daniliuc, Oliver Koch, Bernhard Wünsch
, Org. Biomol. Chem.
, 2021
, 19
, 4082
- Synthesis and pharmacological effects of the enantiomers of the N-phenethyl analogues of the ortho and para e- and f-oxide-bridged phenylmorphans. Josef Zezula, Lisa Singer, Anna K. Przybył, Akihiro Hashimoto, Christina M. Dersch, Richard B. Rothman, Jeffrey Deschamps, Yong Sok Lee, Arthur E. Jacobson, Kenner C. Rice
, Org. Biomol. Chem.
, 2008
, 6
, 2868