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- “All water chemistry” for a concise total synthesis of the novel class anti-anginal drug (RS), (R), and (S)-ranolazine. Damodara N. Kommi, Dinesh Kumar, Asit K. Chakraborti
, Green Chem.
, 2013
, 15
, 756
- Design, synthesis and biological evaluation of AKT inhibitors bearing a piperidin-4-yl appendant. Daoguang Zhang, Dongdong Tong, Dezhi Yang, Jing Sun, Fenghe Zhang, Guisen Zhao
, Med. Chem. Commun.
, 2018
, 9
, 1340
- Structure-based optimization of the piperazino-containing 1,3-disubstituted ureas affording sub-nanomolar inhibitors of soluble epoxide hydrolase. Shao-Xu Huang, Bin Cao, Christophe Morisseau, Yi Jin, Bruce D. Hammock, Ya-Qiu Long
, Med. Chem. Commun.
, 2012
, 3
, 379
- A new strategy for the synthesis of taurine derivatives using the ‘safety-catch’ principle for the protection of sulfonic acids. Sonja Seeberger, Roger J. Griffin, Ian R. Hardcastle, Bernard T. Golding
, Org. Biomol. Chem.
, 2007
, 5
, 132
- Discovery and hit-to-lead evaluation of piperazine amides as selective, state-dependent NaV1.7 inhibitors. Brian A. Sparling, S. Yi, J. Able, H. Bregman, Erin F. DiMauro, R. S. Foti, H. Gao, A. Guzman-Perez, H. Huang, M. Jarosh, T. Kornecook, J. Ligutti, B. C. Milgram, B. D. Moyer, B. Youngblood, V. L. Yu, M. M. Weiss
, Med. Chem. Commun.
, 2017
, 8
, 744
- A systematic exploration of the effects of flexibility and basicity on sigma (σ) receptor binding in a series of substituted diamines. Trent Conroy, Madhura Manohar, Yu Gong, Shane M. Wilkinson, Michael Webster, Brian P. Lieberman, Samuel D. Banister, Tristan A. Reekie, Robert H. Mach, Louis M. Rendina, Michael Kassiou
, Org. Biomol. Chem.
, 2016
, 14
, 9388
- CuI-catalyzed amination of Tröger's base halides: a convenient method for synthesis of unsymmetrical Tröger's bases. Manda Bhaskar Reddy, Potuganti Gal Reddy, Myadaraboina Shailaja, Alla Manjula, Tadikamalla Prabhakar Rao
, RSC Adv.
, 2016
, 6
, 98297
- Identification of a new series of benzothiazinone derivatives with excellent antitubercular activity and improved pharmacokinetic profiles. Lu Xiong, Chao Gao, Yao-Jie Shi, Xin Tao, Juan Rong, Kun-Lin Liu, Cui-Ting Peng, Ning-Yu Wang, Qian Lei, Yi-Wen Zhang, Luo-Ting Yu, Yu-Quan Wei
, RSC Adv.
, 2018
, 8
, 11163
- Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines to develop functionalized ligands to target adenosine receptors: fluorescent ligands as an example. Stephanie Federico, Enrico Margiotta, Silvia Paoletta, Sonja Kachler, Karl-Norbert Klotz, Kenneth A. Jacobson, Giorgia Pastorin, Stefano Moro, Giampiero Spalluto
, Med. Chem. Commun.
, 2019
, 10
, 1094
- Novel fluorescent anthracene–bodipy dyads displaying sensitivity to pH and turn-on behaviour towards Cu(ii) ions. A. Vanessa Saura, M. Isabel Burguete, Francisco Galindo, Santiago V. Luis
, Org. Biomol. Chem.
, 2017
, 15
, 3013