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- Tricyclic xanthine derivatives containing a basic substituent: adenosine receptor affinity and drug-related properties. Michał Załuski, Katarzyna Stanuch, Tadeusz Karcz, Sonja Hinz, Gniewomir Latacz, Ewa Szymańska, Jakub Schabikowski, Agata Doroż-Płonka, Jadwiga Handzlik, Anna Drabczyńska, Christa E. Müller, Katarzyna Kieć-Kononowicz
, Med. Chem. Commun.
, 2018
, 9
, 951
- Studies on enantioselectivity of chiral 4-acetylamino-6-alkyloxy-2-alkylthiopyrimidines acting as antagonists of the human A3 adenosine receptor. Barbara Cosimelli, Giovanni Greco, Sonia Laneri, Ettore Novellino, Antonia Sacchi, Simona Collina, Daniela Rossi, Sandro Cosconati, Elisabetta Barresi, Sabrina Taliani, Maria Letizia Trincavelli, Claudia Martini
, Med. Chem. Commun.
, 2018
, 9
, 81
- Methoxy substituted 2-benzylidene-1-indanone derivatives as A1 and/or A2A AR antagonists for the potential treatment of neurological conditions. Helena D. Janse van Rensburg, Lesetja J. Legoabe, Gisella Terre'Blanche, Mietha M. Van der Walt
, Med. Chem. Commun.
, 2019
, 10
, 300
- Bitopic fluorescent antagonists of the A2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners. Romain Duroux, Antonella Ciancetta, Philip Mannes, Jinha Yu, Shireesha Boyapati, Elizabeth Gizewski, Said Yous, Francisco Ciruela, John A. Auchampach, Zhan-Guo Gao, Kenneth A. Jacobson
, Med. Chem. Commun.
, 2017
, 8
, 1659
- Recent advances in nanomedicine for metabolism-targeted cancer therapy. Jun Da, XinJia Di, YuQi Xie, JiLi Li, LiLi Zhang, YanLan Liu
, Chem. Commun.
, 2024
, 60
, 2442
- Expeditious synthesis and biological evaluation of new C-6 1,2,3-triazole adenosine derivatives A1 receptor
antagonists or agonists. Smitha C. Mathew, Youlet By, Aurélie Berthault, Marie-Alice Virolleaud, Louis Carrega, Gaëlle Chouraqui, Laurent Commeiras, Jocelyne Condo, Mireille Attolini, Anouk Gaudel-Siri, Jean Ruf, Jean Rodriguez, Jean-Luc Parrain, Régis Guieu
, Org. Biomol. Chem.
, 2010
, 8
, 3874
- Structure activity relationship of 2-arylalkynyl-adenine derivatives as human A3 adenosine receptor antagonists. Jinha Yu, Philip Mannes, Young-Hwan Jung, Antonella Ciancetta, Amelia Bitant, David I. Lieberman, Sami Khaznadar, John A. Auchampach, Zhan-Guo Gao, Kenneth A. Jacobson
, Med. Chem. Commun.
, 2018
, 9
, 1920
- Californium-252 plasma desorption mass spectrometry as an aid in the synthesis of a series of adenosine and xanthine conjugates. Kenneth A. Jacobson, Lewis K. Pannell, Kenneth L. Kirk, Henry M. Fales, Edward A. Sokoloski
, J. Chem. Soc., Perkin Trans. 1
, 1986
, 2143
- Application of fluorescence correlation spectroscopy to the measurement of agonist binding to a G-protein coupled receptor at the single cell level. Stephen J. Briddon, Richard J. Middleton, Andrew S. Yates, Michael W. George, Barrie Kellam, Stephen J. Hill
, Faraday Discuss.
, 2004
, 126
, 197
- Stabilised G protein-coupled receptors in structure-based drug design: a case study with adenosine A2A receptor. Stephen P. Andrews, Benjamin Tehan
, Med. Chem. Commun.
, 2013
, 4
, 52