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- Biocatalytic retrosynthesis approaches to d-(2,4,5-trifluorophenyl)alanine, key precursor of the antidiabetic sitagliptin. Fabio Parmeggiani, Arnau Rué Casamajo, Danilo Colombo, Maria Chiara Ghezzi, James L. Galman, Roberto A. Chica, Elisabetta Brenna, Nicholas J. Turner
, Green Chem.
, 2019
, 21
, 4368