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- Targeting Brd4 for cancer therapy: inhibitors and degraders. Yingchao Duan, Yuanyuan Guan, Wenping Qin, Xiaoyu Zhai, Bin Yu, Hongmin Liu
, Med. Chem. Commun.
, 2018
, 9
, 1779
- Discovery of novel trimethoxy-ring BRD4 bromodomain inhibitors: AlphaScreen assay, crystallography and cell-based assay. Zhifeng Chen, Hao Zhang, Shien Liu, Yiqian Xie, Hao Jiang, Wenchao Lu, Heng Xu, Liyan Yue, Yuanyuan Zhang, Hong Ding, Mingyue Zheng, Kunqian Yu, Kaixian Chen, Hualiang Jiang, Cheng Luo
, Med. Chem. Commun.
, 2017
, 8
, 1322
- Structure-based virtual screening of novel, high-affinity BRD4 inhibitors. Charuvaka Muvva, E. R. Azhagiya Singam, S. Sundar Raman, V. Subramanian
, Mol. BioSyst.
, 2014
, 10
, 2384
- Neural tissue engineering: the influence of scaffold surface topography and extracellular matrix microenvironment. Chun-Yi Yang, Wei-Yuan Huang, Liang-Hsin Chen, Nai-Wen Liang, Huan-Chih Wang, Jiaju Lu, Xiumei Wang, Tzu-Wei Wang
, J. Mater. Chem. B
, 2021
, 9
, 567
- Chemical probes and inhibitors of bromodomains outside the BET family. Moses Moustakim, Peter G. K. Clark, Duncan A. Hay, Darren J. Dixon, Paul E. Brennan
, Med. Chem. Commun.
, 2016
, 7
, 2246
- Small molecule-induced cellular conversion. Debojyoti De, Debasish Halder, Injae Shin, Kyeong Kyu Kim
, Chem. Soc. Rev.
, 2017
, 46
, 6241
- Insight into the key interactions of bromodomain inhibitors based on molecular docking, interaction fingerprinting, molecular dynamics and binding free energy calculation. Ting Ran, Zhimin Zhang, Kejun Liu, Yi Lu, Huifang Li, Jinxing Xu, Xiao Xiong, Yanmin Zhang, Anyang Xu, Shuai Lu, Haichun Liu, Tao Lu, Yadong Chen
, Mol. BioSyst.
, 2015
, 11
, 1295
- A chiral-at-metal asymmetric catalyzed vinylogous Michael addition of ortho-methyl aromatic nitro compounds for isoxazole derivative synthesis. Shi-Wu Li, Yu Du, Qiang Kang
, Org. Chem. Front.
, 2019
, 6
, 2775
- Discovery of BET bromodomain inhibitors and their role in target validation. S. Müller, S. Knapp
, Med. Chem. Commun.
, 2014
, 5
, 288
- Fragments in bromodomain drug discovery. Paul Bamborough, Chun-wa Chung
, Med. Chem. Commun.
, 2015
, 6
, 1587