Results
1 -
10 of
19
(Click
here to explore results)
- Aromatic heterocycle galectin-1 interactions for selective single-digit nM affinity ligands. Kristoffer Peterson, Patrick M. Collins, Xiaoli Huang, Barbro Kahl-Knutsson, Sofia Essén, Fredrik R. Zetterberg, Stina Oredsson, Hakon Leffler, Helen Blanchard, Ulf J. Nilsson
, RSC Adv.
, 2018
, 8
, 24913
- Designing interactions by control of protein–ligand complex conformation: tuning arginine–arene interaction geometry for enhanced electrostatic protein–ligand interactions. A.-L. Noresson, O. Aurelius, C. T. Öberg, O. Engström, A. P. Sundin, M. Håkansson, O. Stenström, M. Akke, D. T. Logan, H. Leffler, U. J. Nilsson
, Chem. Sci.
, 2018
, 9
, 1014
- Design and synthesis of novel 3-triazolyl-1-thiogalactosides as galectin-1, -3 and -8 inhibitors. Sjors van Klaveren, Jaka Dernovšek, Žiga Jakopin, Marko Anderluh, Hakon Leffler, Ulf J. Nilsson, Tihomir Tomašič
, RSC Adv.
, 2022
, 12
, 18973
- Symmetric dithiodigalactoside: strategic combination of binding studies and detection of selectivity between a plant toxin and human lectins. Sonsoles Martín-Santamaría, Sabine André, Eliza Buzamet, Rémi Caraballo, Gloria Fernández-Cureses, Maria Morando, João P. Ribeiro, Karla Ramírez-Gualito, Beatriz de Pascual-Teresa, F. Javier Cañada, Margarita Menéndez, Olof Ramström, Jesús Jiménez-Barbero, Dolores Solís, Hans-Joachim Gabius
, Org. Biomol. Chem.
, 2011
, 9
, 5445
- Hybrid ligands with calixarene and thiodigalactoside groups: galectin binding and cytotoxicity. Hao Zhang, Hans Ippel, Michelle C. Miller, Tse J. Wong, Arjan W. Griffioen, Kevin H. Mayo, Roland J. Pieters
, Org. Chem. Front.
, 2019
, 6
, 2981
- Efficient synthesis of a galectin inhibitor clinical candidate (TD139) using a Payne rearrangement/azidation reaction cascade. Jacob St-Gelais, Vincent Denavit, Denis Giguère
, Org. Biomol. Chem.
, 2020
, 18
, 3903
- Tri-isopropylsilyl thioglycosides as masked glycosyl thiol nucleophiles for the synthesis of S-linked glycosides and glyco-conjugates. S. Mandal, U. J. Nilsson
, Org. Biomol. Chem.
, 2014
, 12
, 4816
- Glycomimetics for the inhibition and modulation of lectins. Steffen Leusmann, Petra Ménová, Elena Shanin, Alexander Titz, Christoph Rademacher
, Chem. Soc. Rev.
, 2023
, 52
, 3663
- Substituted polyfluoroaryl interactions with an arginine side chain in galectin-3 are governed by steric-, desolvation and electronic conjugation effects. Rohit Kumar, Kristoffer Peterson, Majda Misini Ignjatović, Hakon Leffler, Ulf Ryde, Ulf J. Nilsson, Derek T. Logan
, Org. Biomol. Chem.
, 2019
, 17
, 1081
- Multivalent glycans for biological and biomedical applications. Yujun Kim, Ji Young Hyun, Injae Shin
, Chem. Soc. Rev.
, 2021
, 50
, 10567