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- Substituent effects on the stability, physicochemical properties and chemical reactivity of nitroimidazole derivatives with potential antiparasitic effect: a computational study. Linda Campos-Fernández, Carolina Barrientos-Salcedo, Edtson E. Herrera Valencia, Rocío Ortiz-Muñiz, Catalina Soriano-Correa
, New J. Chem.
, 2019
, 43
, 11125
- The cubane paradigm in bioactive molecule discovery: further scope, limitations and the cyclooctatetraene complement. Sevan D. Houston, Tyler Fahrenhorst-Jones, Hui Xing, Benjamin A. Chalmers, Melissa L. Sykes, Jeanette E. Stok, Clementina Farfan Soto, Jed M. Burns, Paul V. Bernhardt, James J. De Voss, Glen M. Boyle, Maree T. Smith, John Tsanaktsidis, G. Paul Savage, Vicky M. Avery, Craig M. Williams
, Org. Biomol. Chem.
, 2019
, 17
, 6790
- Synthesis, characterization and biological activities of 3-aryl-1,4-naphthoquinones – green palladium-catalysed Suzuki cross coupling. Aline da R. Louvis, Nayane A. A. Silva, Felipe S. Semaan, Fernando de C. da Silva, Gabriela Saramago, Laís C. S. V. de Souza, Bruno L. A. Ferreira, Helena C. Castro, Juliana P. Salles, André L. A. Souza, Robson X. Faria, Vitor F. Ferreira, Daniela de L. Martins
, New J. Chem.
, 2016
, 40
, 7643
- Imidazoles from nitroallylic acetates and α-bromonitroalkenes with amidines: synthesis and trypanocidal activity studies. Elumalai Gopi, Tarun Kumar, Rubem F. S. Menna-Barreto, Wagner O. Valença, Eufrânio N. da Silva Júnior, Irishi N. N. Namboothiri
, Org. Biomol. Chem.
, 2015
, 13
, 9862
- Quantum mechanical, molecular docking, molecular dynamics, ADMET and antiproliferative activity on Trypanosoma cruzi (Y strain) of chalcone (E)-1-(2-hydroxy-3,4,6-trimethoxyphenyl)-3-(3-nitrophenyl)prop-2-en-1-one derived from a natural product. Maria Geysillene Castro Matos, Leonardo Paes da Silva, Francisco Wagner Queiroz Almeida-Neto, Emanuelle Machado Marinho, Ramon Róseo Paula Pessoa Bezerra de Menezes, Tiago Lima Sampaio, Matheus Nunes da Rocha, Lyanna Rodrigues Ribeiro, Emanuel Paula magalhaes, Alexandre Magno Rodrigues Teixeira, Hélcio Silva dos Santos, Emmanuel Silva Marinho, Pedro de Lima-Neto, Alice Maria Costa Martins, Norberto K. V. Monteiro, Márcia Machado Marinho
, Phys. Chem. Chem. Phys.
, 2022
, 24
, 5052
- Investigation of the antitrypanosomal effects of 2-formyl-8-hydroxyquinoline-derived hydrazones and their antimony(iii) and bismuth(iii) complexes. Ana Paula A. Oliveira, Angel A. Recio-Despaigne, Isabella P. Ferreira, Renata Diniz, Karoline A. F. Sousa, Tanira M. Bastos, Milena B. Pereira Soares, Diogo Rodrigo M. Moreira, Heloisa Beraldo
, New J. Chem.
, 2019
, 43
, 18996
- Selenosemicarbazones as potent cruzipain inhibitors and their antiparasitic properties against Trypanosoma
cruzi. Chiara Pizzo, Paula Faral-Tello, Gustavo Salinas, Martín Fló, Carlos Robello, Peter Wipf, S. Graciela Mahler
, Med. Chem. Commun.
, 2012
, 3
, 362
- Development of new dinuclear Fe(iii) coordination compounds with in vitro nanomolar antitrypanosomal activity. Felipe Figueirôa Moreira, Juliana de Araujo Portes, Nathália Florência Barros Azeredo, Christiane Fernandes, Adolfo Horn, Cristina Pinheiro Santiago, Bruna Barriquel Segat, Giovanni Finoto Caramori, Letícia Maria Pequeno Madureira, Dalber Ruben Sanchez Candela, Marcelo Monteiro Marques, Jackson Antônio Lamounier Camargos Resende, Wanderley de Souza, Renato Augusto DaMatta, Sergio Henrique Seabra
, Dalton Trans.
, 2021
, 50
, 12242
- Curcumin inspired synthesis of unsymmetrical diarylpentanoids with highly potent anti-parasitic activities: in silico studies and DFT-based stereochemical calculation. Zia Ud Din, Alef dos Santos, Marilia Almeida Trapp, Danielle Lazarin-Bidóia, Francielle Pelegrin Garcia, Francieli Peron, Celso Vataru Nakamura, Edson Rodrigues-Filho
, Med. Chem. Commun.
, 2016
, 7
, 820
- Antiprotozoal activity of dehydroabietic acid derivatives against Leishmania donovani and Trypanosoma cruzi. Mikko Vahermo, Sara Krogerus, Abdelmajeed Nasereddin, Marcel Kaiser, Reto Brun, Charles L. Jaffe, Jari Yli-Kauhaluoma, Vânia M. Moreira
, Med. Chem. Commun.
, 2016
, 7
, 457