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- Chemical probes and inhibitors of bromodomains outside the BET family. Moses Moustakim, Peter G. K. Clark, Duncan A. Hay, Darren J. Dixon, Paul E. Brennan
, Med. Chem. Commun.
, 2016
, 7
, 2246
- Cation–π interactions in CREBBP bromodomain inhibition: an electrostatic model for small-molecule binding affinity and selectivity. Wilian A. Cortopassi, Kiran Kumar, Robert S. Paton
, Org. Biomol. Chem.
, 2016
, 14
, 10926
- Classical molecular dynamics and metadynamics simulations decipher the mechanism of CBP30 selectively inhibiting CBP/p300 bromodomains. Qianqian Wang, Xiaoli An, Jiahui Xu, Yuwei Wang, Liang Liu, Elaine Lai-Han Leung, Xiaojun Yao
, Org. Biomol. Chem.
, 2018
, 16
, 6521
- A poised fragment library enables rapid synthetic expansion yielding the first reported inhibitors of PHIP(2), an atypical bromodomain. Oakley B. Cox, Tobias Krojer, Patrick Collins, Octovia Monteiro, Romain Talon, Anthony Bradley, Oleg Fedorov, Jahangir Amin, Brian D. Marsden, John Spencer, Frank von Delft, Paul E. Brennan
, Chem. Sci.
, 2016
, 7
, 2322