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- Synthesis and configuration determination of all enantiopure stereoisomers of the melatonin receptor ligand
4-phenyl-2-propionamidotetralin using an expedient optical resolution of 4-phenyl-2-tetralone. Simone Lucarini, Silvia Bartolucci, Annalida Bedini, Giuseppe Gatti, Pierfrancesco Orlando, Giovanni Piersanti, Gilberto Spadoni
, Org. Biomol. Chem.
, 2012
, 10
, 305
- An improved synthesis of
cis-4-phenyl-2-propionamidotetralin (4-P-PDOT): a selective MT2melatonin receptor antagonist. Simone Lucarini, Annalida Bedini, Gilberto Spadoni, Giovanni Piersanti
, Org. Biomol. Chem.
, 2008
, 6
, 147
- An efficient route to highly enantioenriched tetrahydroazulenes and β-tetralones by desymmetrization reactions of δ,δ-diaryldiazoaceto-acetates. Yuxiao Liu, Yongming Deng, Peter Y. Zavalij, Renhua Liu, Michael P. Doyle
, Chem. Commun.
, 2015
, 51
, 565
- Design, synthesis, and biological evaluation of a new class of MT2-selective agonists. Xuan Zhang, Zhilong Wang, Qingqing Huang, Yu Luo, Xin Xie, Wei Lu
, RSC Adv.
, 2014
, 4
, 25871
- N1-linked melatonin dimers as bivalent ligands targeting dimeric melatonin receptors. Anne-Sophie Journé, Samy A. M. Habib, Bala R. Dodda, Mina N. F. Morcos, Mirna S. Sadek, Sarah A. A. Tadros, Paula A. Witt-Enderby, Ralf Jockers, Darius P. Zlotos
, Med. Chem. Commun.
, 2014
, 5
, 792