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- Design, synthesis and biological evaluation of pyrazolo[3,4-b]pyridine derivatives as TRK inhibitors. Nian Liu, Xin Wang, Qinglin Fu, Qiaohua Qin, Tianxiao Wu, Ruicheng Lv, Dongmei Zhao, Maosheng Cheng
, RSC Med. Chem.
, 2023
, 14
, 85
- Pyrazole-containing pharmaceuticals: target, pharmacological activity, and their SAR studies. Guangchen Li, Yifu Cheng, Chi Han, Chun Song, Niu Huang, Yunfei Du
, RSC Med. Chem.
, 2022
, 13
, 1300
- Kinase inhibitor macrocycles: a perspective on limiting conformational flexibility when targeting the kinome with small molecules. Baku Acharya, Debasmita Saha, Daniel Armstrong, Baha'a Jabali, Maha Hanafi, Alan Herrera-Rueda, Naga Rajiv Lakkaniga, Brendan Frett
, RSC Med. Chem.
, 2024
, 15
, 399
- Biocatalytic reductive aminations with NAD(P)H-dependent enzymes: enzyme discovery, engineering and synthetic applications. Bo Yuan, Dameng Yang, Ge Qu, Nicholas J. Turner, Zhoutong Sun
, Chem. Soc. Rev.
, 2024
, 53
, 227
- Discovery of Cobimetinib as a novel A-FABP inhibitor using machine learning and molecular docking-based virtual screening. Shilun Yang, Simeng Li, Junlei Chang
, RSC Adv.
, 2022
, 12
, 13500
- Computational design of an imine reductase: mechanism-guided stereoselectivity reversion and interface stabilization. Kai Wu, Jinrong Yan, Qinde Liu, Xiaojing Wang, Piaoru Wu, Yiyang Cao, Xiuhong Lu, Yixin Xu, Junhai Huang, Lei Shao
, Chem. Sci.
, 2024
, 15
, 1431
- A sumanene-containing magnetic nanoadsorbent for the removal of caesium salts from aqueous solutions. Artur Kasprzak, Magdalena Matczuk, Hidehiro Sakurai
, Chem. Commun.
, 2023
, 59
, 9591
- Synthetic inhibitor leads of human tropomyosin receptor kinase A (hTrkA). Govindan Subramanian, Rajendran Vairagoundar, Scott J. Bowen, Nicole Roush, Theresa Zachary, Christopher Javens, Tracey Williams, Ann Janssen, Andrea Gonzales
, RSC Med. Chem.
, 2020
, 11
, 370
- A soluble iron(ii)-phthalocyanine-catalyzed intramolecular C(sp3)–H amination with alkyl azides. Tingjie You, Si-Hao Zeng, Jianqiang Fan, Liangliang Wu, Fangyuan Kang, Yungen Liu, Chi-Ming Che
, Chem. Commun.
, 2021
, 57
, 10711
- Asymmetric organocatalysis: an enabling technology for medicinal chemistry. Bo Han, Xiang-Hong He, Yan-Qing Liu, Gu He, Cheng Peng, Jun-Long Li
, Chem. Soc. Rev.
, 2021
, 50
, 1522