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- New pyrazolo[3,4-b]pyridones as selective A1 adenosine receptor antagonists: synthesis, biological evaluation and molecular modelling studies. Paola Fossa, Marco Pestarino, Giulia Menozzi, Luisa Mosti, Silvia Schenone, Angelo Ranise, Francesco Bondavalli, M. Letizia Trincavelli, Antonio Lucacchini, Claudia Martini
, Org. Biomol. Chem.
, 2005
, 3
, 2262
- Regio- and stereoselective synthesis of truncated 3′-aminocarbanucleosides and their binding affinity at the A3
adenosine
receptor. Mun Ju Choi, Girish Chandra, Hyuk Woo Lee, Xiyan Hou, Won Jun Choi, Khai Phan, Kenneth A. Jacobson, Lak Shin Jeong
, Org. Biomol. Chem.
, 2011
, 9
, 6955
- Pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidines to develop functionalized ligands to target adenosine receptors: fluorescent ligands as an example. Stephanie Federico, Enrico Margiotta, Silvia Paoletta, Sonja Kachler, Karl-Norbert Klotz, Kenneth A. Jacobson, Giorgia Pastorin, Stefano Moro, Giampiero Spalluto
, Med. Chem. Commun.
, 2019
, 10
, 1094
- Ligand design by targeting a binding site water. Pierre Matricon, R. Rama Suresh, Zhan-Guo Gao, Nicolas Panel, Kenneth A. Jacobson, Jens Carlsson
, Chem. Sci.
, 2021
, 12
, 960
- Demystifying the three dimensional structure of G protein-coupled receptors (GPCRs) with the aid of molecular modeling. Stefano Moro, Francesca Deflorian, Giampiero Spalluto, Giorgia Pastorin, Barbara Cacciari, Soo-Kyung Kim, Kenneth A. Jacobson
, Chem. Commun.
, 2003
, 2949
- Structure activity relationship of 2-arylalkynyl-adenine derivatives as human A3 adenosine receptor antagonists. Jinha Yu, Philip Mannes, Young-Hwan Jung, Antonella Ciancetta, Amelia Bitant, David I. Lieberman, Sami Khaznadar, John A. Auchampach, Zhan-Guo Gao, Kenneth A. Jacobson
, Med. Chem. Commun.
, 2018
, 9
, 1920
- Convergent synthesis of 2-thioether-substituted (N)-methanocarba-adenosines as purine receptor agonists. R. Rama Suresh, Russell B. Poe, Baorui Lin, Kexin Lv, Ryan G. Campbell, Zhan-Guo Gao, Theodore E. Liston, Kiran S. Toti, Kenneth A. Jacobson
, RSC Adv.
, 2021
, 11
, 27369
- Bitopic fluorescent antagonists of the A2A adenosine receptor based on pyrazolo[4,3-e][1,2,4]triazolo[1,5-c]pyrimidin-5-amine functionalized congeners. Romain Duroux, Antonella Ciancetta, Philip Mannes, Jinha Yu, Shireesha Boyapati, Elizabeth Gizewski, Said Yous, Francisco Ciruela, John A. Auchampach, Zhan-Guo Gao, Kenneth A. Jacobson
, Med. Chem. Commun.
, 2017
, 8
, 1659