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- Covalent inhibitors: a rational approach to drug discovery. Fandi Sutanto, Markella Konstantinidou, Alexander Dömling
, RSC Med. Chem.
, 2020
, 11
, 876
- Highly enantioselective Rh-catalyzed asymmetric reductive dearomatization of multi-nitrogen polycyclic pyrazolo[1,5-a]pyrimidines. Chaochao Xie, Guiying Xiao, Qianling Guo, Xiaoxue Wu, Guofu Zi, Wanjian Ding, Guohua Hou
, Chem. Sci.
, 2023
, 14
, 9048
- Pyrazole-containing pharmaceuticals: target, pharmacological activity, and their SAR studies. Guangchen Li, Yifu Cheng, Chi Han, Chun Song, Niu Huang, Yunfei Du
, RSC Med. Chem.
, 2022
, 13
, 1300
- Advanced approaches of developing targeted covalent drugs. Conghao Gai, Suzannah J. Harnor, Shihao Zhang, Céline Cano, Chunlin Zhuang, Qingjie Zhao
, RSC Med. Chem.
, 2022
, 13
, 1460
- A primer on harnessing non-enzymatic post-translational modifications for drug design. Marcus J. C. Long, Phillippe Ly, Yimon Aye
, RSC Med. Chem.
, 2021
, 12
, 1797
- Recent advances in the development of covalent inhibitors. Hyunsoo Kim, Yoon Soo Hwang, Mingi Kim, Seung Bum Park
, RSC Med. Chem.
, 2021
, 12
, 1037
- A mechanistic study of thiol addition to N-acryloylpiperidine. Sarah K. I. Watt, Janique G. Charlebois, Christopher N. Rowley, Jeffrey W. Keillor
, Org. Biomol. Chem.
, 2023
, 21
, 2204
- Insights into the medicinal chemistry of heterocycles integrated with a pyrazolo[1,5-a]pyrimidine scaffold. Mohamed M. Hammouda, Hatem E. Gaffer, Khaled M. Elattar
, RSC Med. Chem.
, 2022
, 13
, 1150
- Coumarin–carbazole based functionalized pyrazolines: synthesis, characterization, anticancer investigation and molecular docking. Mrugesh Patel, Nilesh Pandey, Jignesh Timaniya, Paranjay Parikh, Alex Chauhan, Neeraj Jain, Kaushal Patel
, RSC Adv.
, 2021
, 11
, 27627
- Mechanism of covalent binding of ibrutinib to Bruton's tyrosine kinase revealed by QM/MM calculations. Angus T. Voice, Gary Tresadern, Rebecca M. Twidale, Herman van Vlijmen, Adrian J. Mulholland
, Chem. Sci.
, 2021
, 12
, 5511