Results
1 -
3 of
3
(Click
here to explore results)
- Kinase inhibitor macrocycles: a perspective on limiting conformational flexibility when targeting the kinome with small molecules. Baku Acharya, Debasmita Saha, Daniel Armstrong, Baha'a Jabali, Maha Hanafi, Alan Herrera-Rueda, Naga Rajiv Lakkaniga, Brendan Frett
, RSC Med. Chem.
, 2024
, 15
, 399
- Design, synthesis and biological evaluation of pyrazolo[3,4-b]pyridine derivatives as TRK inhibitors. Nian Liu, Xin Wang, Qinglin Fu, Qiaohua Qin, Tianxiao Wu, Ruicheng Lv, Dongmei Zhao, Maosheng Cheng
, RSC Med. Chem.
, 2023
, 14
, 85
- Pyrazole-containing pharmaceuticals: target, pharmacological activity, and their SAR studies. Guangchen Li, Yifu Cheng, Chi Han, Chun Song, Niu Huang, Yunfei Du
, RSC Med. Chem.
, 2022
, 13
, 1300