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61Turlington M; Noetzel MJ; Chun A; Bridges TM; Daniels JS; Jones C; Niswender CM; Meiler J; Conn PJ; Lindsley CW; Stauffer SR; Zhou Y; Gogliotti RD; Nguyen ED; Gregory KJ; Vinson PN; Rook JM; Gogi KK; Xiang Z.
Exploration of allosteric agonism structure-activity relationships within an acetylene series of metabotropic glutamate receptor 5 (mGlu5) positive allosteric modulators (PAMs): discovery of 5-((3-fluorophenyl)ethynyl)-N-(3-methyloxetan-3-yl)picolinamide (ML254)., Journal of medicinal chemistry Fiorino F; Severino B; Magli E; Caliendo G; Perissutti E; Frecentese F; Esposito A; Incisivo GM; Ciano A; Massarelli P; Nencini C; Santagada V.
New potent 5-HT(2A) receptor ligands containing an N'-cyanopicolinamidine nucleus: Synthesis and in?vitro pharmacological evaluation., European journal of medicinal chemistry Ryu JH; Kim S; Han HY; Son HJ; Lee HJ; Shin YA; Kim JS; Park HG.
Synthesis and biological evaluation of picolinamides as potent inhibitors of 11?-hydroxysteroid dehydrogenase type 1 (11?-HSD1)., Bioorganic & medicinal chemistry letters