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1Vilums M; Zweemer AJ; Yu Z; Brussee J; Stamos D; Saunders J; Heitman LH; Ijzerman AP; de Vries H; Hillger JM; Wapenaar H; Bollen IA; Barmare F; Gross R; Clemens J; Krenitsky P.
Structure-kinetic relationships--an overlooked parameter in hit-to-lead optimization: a case of cyclopentylamines as chemokine receptor 2 antagonists., Journal of medicinal chemistry