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1Hayashi Shigeo, Nakata Eriko, Morita Asato, Mizuno Kunihiko, Yamamura Kenzo, Kato Aki, Ohashi Katsuyo.
Discovery of {1-[4-(2-{hexahydropyrrolo[3,4-c]pyrrol-2(1H)-yl}-1H-benzimidazol-1-yl)piperidin-1-yl]cyclooctyl}methanol, systemically potent novel non-peptide agonist of nociceptin/orphanin FQ receptor as analgesic for the treatment of neuropathic pain: Design, synthesis, and structure–activity relationships, Bioorganic & Medicinal Chemistry, 2010