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1539Lu H; Silverman RB.
Fluorinated conformationally restricted gamma-aminobutyric acid aminotransferase inhibitors., Journal of medicinal chemistry Pan Y; Gerasimov MR; Kvist T; Brodie JD; Schiffer WK; Dewey SL; Miller SR; Silverman RB; Wellendorph P; Madsen KK; Pera E; Lee H; Schousboe A; Chebib M; Br?uner-Osborne H; Craft CM.
(1S, 3S)-3-amino-4-difluoromethylenyl-1-cyclopentanoic acid (CPP-115), a potent ?-aminobutyric acid aminotransferase inactivator for the treatment of cocaine addiction., Journal of medicinal chemistry Pan Y; Qiu J; Silverman RB.
Design, synthesis, and biological activity of a difluoro-substituted, conformationally rigid vigabatrin analogue as a potent gamma-aminobutyric acid aminotransferase inhibitor., Journal of medicinal chemistry Juncosa JI Jr; Groves AP; Xia G; Silverman RB.
Probing the steric requirements of the ?-aminobutyric acid aminotransferase active site with fluorinated analogues of vigabatrin., Bioorganic & medicinal chemistry