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2McElroy, Timothy; Thomas, James B.; Brine, George A.; Navarro, Hernán A.; Deschamps, Jeffrey; Carroll, F. Ivy, Synthesis 2008, 943-947.
A Practical Synthesis of the Kappa Opioid Receptor Selective Agonist (+)-5R,7S,8S-N-Methyl-N-[7-(1-pyrrolidinyl)-1-oxospiro[4,5]dec-8-yl]ben­zeneacetamide (U69,593), Synthesis