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2Dow Robert L., Carpino Philip A., Hadcock John R., Black Shawn C., Iredale Philip A., DaSilva-Jardine Paul, Schneider Steven R., Paight Ernest S., Griffith David A., Scott Dennis O., O’Connor Rebecca E., Nduaka Chudy I..
Discovery of 2-(2-Chlorophenyl)-3-(4-chlorophenyl)-7-(2,2-difluoropropyl)-6,7-dihydro-2H-pyrazolo[3,4-f][1,4]oxazepin-8(5H)-one (PF-514273), a Novel, Bicyclic Lactam-Based Cannabinoid-1 Receptor Antagonist for the Treatment of Obesity, Journal of Medicinal Chemistry, 2009