ChemSpider 2D Image | Rimcazole hydrochloride | C21H29Cl2N3

Rimcazole hydrochloride

  • Molecular FormulaC21H29Cl2N3
  • Average mass394.381 Da
  • Monoisotopic mass393.173859 Da
  • ChemSpider ID48220

  • defined stereocentres - 2 of 2 defined stereocentres

More details:

Validated by Experts, Validated by Users, Non-Validated, Removed by Users

2XAC11FCQ4
75859-03-9 [RN]
9-{3-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]propyl}-9H-carbazoldihydrochlorid [German] [ACD/IUPAC Name]
9-{3-[(3R,5S)-3,5-Dimethyl-1-piperazinyl]propyl}-9H-carbazole dihydrochloride [ACD/IUPAC Name]
9-{3-[(3R,5S)-3,5-Diméthyl-1-pipérazinyl]propyl}-9H-carbazole, dichlorhydrate [French] [ACD/IUPAC Name]
9-{3-[(3R,5S)-3,5-Dimethylpiperazin-1-yl]propyl}-9H-carbazole dihydrochloride
9H-Carbazole, 9-[3-[(3R,5S)-3,5-dimethyl-1-piperazinyl]propyl]-, hydrochloride (1:2) [ACD/Index Name]
Rimcazole dihydrochloride
Rimcazole hydrochloride [USAN]
[75859-03-9] [RN]
More...

Validated by Experts, Validated by Users, Non-Validated, Removed by Users

D02684 [DBID]
  • Experimental Physico-chemical Properties
  • Miscellaneous

    • Bio Activity:

      ?2 antagonist. Also DAT inhibitor Tocris Bioscience 1497
      Antagonist at ? receptors (IC50 values are 1480 and 386 nM at ?1 and ?2 receptors respectively). Also binds to the dopamine transporter (IC50 = 57.6 nM) and inhibits dopamine uptake. Reduces the stimu latory effects of cocaine in vivo. Tocris Bioscience 1497
      Antagonist at ? receptors (IC50 values are 1480 and 386 nM at ?1 and ?2 receptors respectively). Also binds to the dopamine transporter (IC50 = 57.6 nM) and inhibits dopamine uptake. Reduces the stimulatory effects of cocaine in vivo. Tocris Bioscience 1497
      Antagonist at sigma receptors (IC50 values are 1480 and 386 nM at sigma1 and sigma2 receptors respectively). Also binds to the dopamine transporter (IC50 = 57.6 nM) and inhibits dopamine uptake. Reduces the stimulatory effects of cocaine in vivo. Tocris Bioscience 1497
      Other Pharmacology Tocris Bioscience 1497
      Sigma Receptors Tocris Bioscience 1497
      sigma2 antagonist. Also DAT inhibitor Tocris Bioscience 1497
      Sigma2 Receptors Tocris Bioscience 1497

Predicted data is generated using the ACD/Labs Percepta Platform - PhysChem Module, version: 14.00

No predicted properties have been calculated for this compound.

Click to predict properties on the Chemicalize site


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