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- Pyrimethamine analogs as strong inhibitors of double and quadruple mutants of dihydrofolate reductase in human malaria parasites. Alireza Sardarian, Kenneth T. Douglas, Martin Read, Paul F. G. Sims, John E. Hyde, Penchit Chitnumsub, Rachada Sirawaraporn, Worachart Sirawaraporn
, Org. Biomol. Chem.
, 2003
, 1
, 960
- Revitalizing antifolates through understanding mechanisms that govern susceptibility and resistance. Shannon Lynn Kordus, Anthony David Baughn
, Med. Chem. Commun.
, 2019
, 10
, 880
- Triazine–pyrimidine based molecular hybrids: synthesis, docking studies and evaluation of antimalarial activity. Deepak Kumar, Shabana I. Khan, Prija Ponnan, Diwan S. Rawat
, New J. Chem.
, 2014
, 38
, 5087
- Highly active 4-aminoquinoline–pyrimidine based molecular hybrids as potential next generation antimalarial agents. Sunny Manohar, V. Satya Pavan, Dale Taylor, Deepak Kumar, Prija Ponnan, Lubbe Wiesner, Diwan S. Rawat
, RSC Adv.
, 2015
, 5
, 28171
- Chloroquinoline–acetamide hybrids: a promising series of potential antiprotozoal agents. Afreen Inam, Robyn L. Van Zyl, Natasha J. van Vuuren, Chien-Teng Chen, Fernando Avecilla, Subhash M. Agarwal, Amir Azam
, RSC Adv.
, 2015
, 5
, 48368
- Design, synthesis and biological evaluation of 6-aryl-1,6-dihydro-1,3,5-triazine-2,4-diamines as antiplasmodial antifolates. Anna C. U. Lourens, David Gravestock, Robyn L. van Zyl, Heinrich C. Hoppe, Natasha Kolesnikova, Supannee Taweechai, Yongyuth Yuthavong, Sumalee Kamchonwongpaisan, Amanda L. Rousseau
, Org. Biomol. Chem.
, 2016
, 14
, 7899
- Thienopyrimidine sulphonamide hybrids: design, synthesis, antiprotozoal activity and molecular docking studies. Saadia Leeza Zaidi, Subhash M. Agarwal, Porntip Chavalitshewinkoon-Petmitr, Thidarat Suksangpleng, Kamal Ahmad, Fernando Avecilla, Amir Azam
, RSC Adv.
, 2016
, 6
, 90371
- Antimalarial activity and docking studies of novel bi-functional hybrids derived from 4-aminoquinoline and 1,3,5-triazine against wild and mutant malaria parasites as pf-DHFR inhibitor. Hans Raj Bhat, Udaya Pratap Singh, Prashant Gahtori, Surajit Kumar Ghosh, Kabita Gogoi, Anil Prakash, Ramendra K. Singh
, RSC Adv.
, 2013
, 3
, 2942
- Synthesis, antimalarial activity, heme binding and docking studies of 4-aminoquinoline–pyrimidine based molecular hybrids. Deepak Kumar, Shabana I. Khan, Babu L. Tekwani, Prija Ponnan, Diwan S. Rawat
, RSC Adv.
, 2014
, 4
, 63655
- 4-Aminoquinoline-pyrimidine-aminoalkanols: synthesis, in vitro antimalarial activity, docking studies and ADME predictions. Mohit Tripathi, Shabana I. Khan, Anuj Thakur, Prija Ponnan, Diwan S. Rawat
, New J. Chem.
, 2015
, 39
, 3474