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- Chemogenomics for drug discovery: clinical molecules from open access chemical probes. Robert B. A. Quinlan, Paul E. Brennan
, RSC Chem. Biol.
, 2021
, 2
, 759
- Targeting Brd4 for cancer therapy: inhibitors and degraders. Yingchao Duan, Yuanyuan Guan, Wenping Qin, Xiaoyu Zhai, Bin Yu, Hongmin Liu
, Med. Chem. Commun.
, 2018
, 9
, 1779
- Deciphering the mechanisms of selective inhibition for the tandem BD1/BD2 in the BET-bromodomain family. Chunyan Cheng, Hongjuan Diao, Fan Zhang, Yongheng Wang, Kai Wang, Ruibo Wu
, Phys. Chem. Chem. Phys.
, 2017
, 19
, 23934
- Enzyme-responsive micellar JQ1 induces enhanced BET protein inhibition and immunotherapy of malignant tumors. Zhenqi Zhang, Qiang Zhang, Jiguo Xie, Zhiyuan Zhong, Chao Deng
, Biomater. Sci.
, 2021
, 9
, 6915
- Importance of a crystalline water network in docking-based virtual screening: a case study of BRD4. Haiyang Zhong, Zhe Wang, Xuwen Wang, Hui Liu, Dan Li, Huanxiang Liu, Xiaojun Yao, Tingjun Hou
, Phys. Chem. Chem. Phys.
, 2019
, 21
, 25276
- Analysis of physicochemical properties of protein–protein interaction modulators suggests stronger alignment with the “rule of five”. Jia Truong, Ashwin George, Jessica K. Holien
, RSC Med. Chem.
, 2021
, 12
, 1731
- Tricyclic 2-benzazepines obtained via an unexpected cyclization involving nitrilium ylides. Anna Inyutina, Dmitry Dar'in, Grigory Kantin, Mikhail Krasavin
, Org. Biomol. Chem.
, 2021
, 19
, 5068
- Chemically induced degradation of epigenetic targets. Md Kabir, Xufen Yu, H. Ümit Kaniskan, Jian Jin
, Chem. Soc. Rev.
, 2023
, 52
, 4313
- The binding mechanism of NHWD-870 to bromodomain-containing protein 4 based on molecular dynamics simulations and free energy calculation. Mingsong Shi, Jun He, Tiantian Weng, Na Shi, Wenyan Qi, Yong Guo, Tao Chen, Lijuan Chen, Dingguo Xu
, Phys. Chem. Chem. Phys.
, 2022
, 24
, 5125
- Bromodomain and extraterminal protein-targeted probe enables tumour visualisation in vivo using positron emission tomography. Catherine G. Fitzgerald Dickmann, Alexander F. McDonald, Nhi Huynh, Angela Rigopoulos, Zhanqi Liu, Nancy Guo, Laura D. Osellame, Michael A. Gorman, Michael W. Parker, Hui K. Gan, Andrew M. Scott, Uwe Ackermann, Ingrid J. G. Burvenich, Jonathan M. White
, Chem. Commun.
, 2023
, 59
, 3126