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Small-molecule inhibitors of HIF-PHD2: a valid strategy to renal anemia treatment in clinical therapy . Yue Wu, Nan Wang, Yonghua Lei, Tianhan Hu, Qidong You, Xiaojin Zhang
, Med. Chem. Commun.
, 2016
, 7
, 1271
Molecular and cellular mechanisms of HIF prolyl hydroxylase inhibitors in clinical trials . Tzu-Lan Yeh, Thomas M. Leissing, Martine I. Abboud, Cyrille C. Thinnes, Onur Atasoylu, James P. Holt-Martyn, Dong Zhang, Anthony Tumber, Kerstin Lippl, Christopher T. Lohans, Ivanhoe K. H. Leung, Helen Morcrette, Ian J. Clifton, Timothy D. W. Claridge, Akane Kawamura, Emily Flashman, Xin Lu, Peter J. Ratcliffe, Rasheduzzaman Chowdhury, Christopher W. Pugh, Christopher J. Schofield
, Chem. Sci.
, 2017
, 8
, 7651
A small-molecule probe for monitoring binding to prolyl hydroxylase domain 2 by fluorescence polarisation . Zhihong Li, Shuai Zhen, Kaijun Su, Anthony Tumber, Quanwei Yu, Ying Dong, Michael McDonough, Christopher J. Schofield, Xiaojin Zhang
, Chem. Commun.
, 2020
, 56
, 14199
Structure-guided optimisation of N -hydroxythiazole-derived inhibitors of factor inhibiting hypoxia-inducible factor-α . Thomas P. Corner, Ryan Z. R. Teo, Yue Wu, Eidarus Salah, Yu Nakashima, Giorgia Fiorini, Anthony Tumber, Amelia Brasnett, James P. Holt-Martyn, William D. Figg, Xiaojin Zhang, Lennart Brewitz, Christopher J. Schofield
, Chem. Sci.
, 2023
, 14
, 12098
Kinetic and inhibition studies on human Jumonji-C (JmjC) domain-containing protein 5 . Anthony Tumber, Eidarus Salah, Lennart Brewitz, Thomas P. Corner, Christopher J. Schofield
, RSC Chem. Biol.
, 2023
, 4
, 399
Studies on spiro[4.5]decanone prolyl hydroxylase domain inhibitors . James P. Holt-Martyn, Anthony Tumber, Mohammed Z. Rahman, Kerstin Lippl, William Figg, Michael A. McDonough, Rasheduzzaman Chowdhury, Christopher J. Schofield
, Med. Chem. Commun.
, 2019
, 10
, 500
Evaluating and clustering retrosynthesis pathways with learned strategy . Yiming Mo, Yanfei Guan, Pritha Verma, Jiang Guo, Mike E. Fortunato, Zhaohong Lu, Connor W. Coley, Klavs F. Jensen
, Chem. Sci.
, 2021
, 12
, 1469
A comprehensive and high-throughput screening method for multiple prohibited substances by UPLC-QE Plus-HRMS and HPLC-QQQ-MS in human urine for doping control . Yunxi Liu, Tianyu Dong, Kuan Yan, Zhanliang Wang, Genye He, Yufeng Zhang, Congcong Ma, Lu Liu, Wei Chang, Lisi Zhang
, Anal. Methods
, 2023
, 15
, 3206