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- Pyridazinone derivatives as potential anti-inflammatory agents: synthesis and biological evaluation as PDE4 inhibitors. Ingrid Allart-Simon, Aurélie Moniot, Nicolo Bisi, Miguel Ponce-Vargas, Sandra Audonnet, Marie Laronze-Cochard, Janos Sapi, Eric Hénon, Frédéric Velard, Stéphane Gérard
, RSC Med. Chem.
, 2021
, 12
, 584
- Diastereoselective synthesis and profiling of bicyclic imidazolidinone derivatives bearing a difluoromethylated catechol unit as potent phosphodiesterase 4 inhibitors. Valentin S. Dorokhov, Ivan S. Golovanov, Vladimir A. Tartakovsky, Alexey Yu. Sukhorukov, Sema L. Ioffe
, Org. Biomol. Chem.
, 2018
, 16
, 6900
- Generation of difluorocarbenes and introduction of fluorinated one carbon units into carbonyl and related compounds. Kohei Fuchibe, Junji Ichikawa
, Chem. Commun.
, 2023
, 59
, 2532
- Microwave-assisted synthesis of potent PDE7 inhibitors containing a thienopyrimidin-4-amine scaffold. Ana I. Sánchez, Ricardo Meneses, José M. Mínguez, Araceli Núñez, Rafael R. Castillo, Fabiana Filace, Carolina Burgos, Juan J. Vaquero, Julio Álvarez-Builla, Alvaro Cortés-Cabrera, Federico Gago, Emma Terricabras, Víctor Segarra
, Org. Biomol. Chem.
, 2014
, 12
, 4233
- Computational analyses of mechanism of action (MoA): data, methods and integration. Maria-Anna Trapotsi, Layla Hosseini-Gerami, Andreas Bender
, RSC Chem. Biol.
, 2022
, 3
, 170
- Selective inhibitors of phosphodiesterases: therapeutic promise for neurodegenerative disorders. Tarana Umar, Nasimul Hoda
, Med. Chem. Commun.
, 2015
, 6
, 2063
- Anthranilic acid-based inhibitors of phosphodiesterase: Design, synthesis, and bioactive evaluation. Yih-Dih Cheng, Tsong-Long Hwang, Han-Hsiang Wang, Tai-Long Pan, Chin-Chung Wu, Wen-Yi Chang, Yi-Ting Liu, Tzu-Chi Chu, Pei-Wen Hsieh
, Org. Biomol. Chem.
, 2011
, 9
, 7113