Results
1 -
1 of
1Di Fabio Romano, Griffante Cristiana, Alvaro Giuseppe, Pentassuglia Giorgio, Pizzi Domenica A., Donati Daniele, Rossi Tino, Guercio Giuseppe, Mattioli Mario, Cimarosti Zadeo, Marchioro Carla, Provera Stefano, Zonzini Laura, Montanari Dino, Melotto Sergio, Gerrard Philip A., Trist David G., Ratti Emiliangelo, Corsi Mauro.
Discovery Process and Pharmacological Characterization of 2-(S)-(4-Fluoro-2-methylphenyl)piperazine-1-carboxylic Acid [1-(R)-(3,5-Bis-trifluoromethylphenyl)ethyl]methylamide (Vestipitant) as a Potent, Selective, and Orally Active NK1Receptor Antagonist, Journal of Medicinal Chemistry, 2009