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1Das Jagabandhu, Chen Ping, Norris Derek, Padmanabha Ramesh, Lin James, Moquin Robert V., Shen Zhongqi, Cook Lynda S., Doweyko Arthur M., Pitt Sidney, Pang Suhong, Shen Ding Ren, Fang Qiong, de Fex Henry F., McIntyre Kim W., Shuster David J., Gillooly Kathleen M., Behnia Kamelia, Schieven Gary L., Wityak John, Barrish Joel C..
2-Aminothiazole as a Novel Kinase Inhibitor Template. Structure−Activity Relationship Studies toward the Discovery ofN-(2-Chloro-6-methylphenyl)-2-[[6-[4-(2-hydroxyethyl)-1- piperazinyl)]-2-methyl-4-pyrimidinyl]amino)]-1,3-thiazole-5-carboxamide (Dasatinib, BMS-354825) as a Potentpan-Src Kinase Inhibitor, Journal of Medicinal Chemistry, 2006