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3Sonoshita et al.
A whole-animal platform to advance a clinical kinase inhibitor into new disease space.
Nature Chemical Biology, doi: 10.1038/nchembio.2556, published online 22 January 2018 Kleemann, A.; Engel, J.; Kutscher, B.; Reichert, D., Pharmaceutical Substances [Online], Thieme: Stuttgart, (2014)..
Trametinib, Pharmaceutical Substances Guan Longfei, Yang Hongbin, Cai Yingchun, Sun Lixia, Di Peiwen, Li Weihua, Liu Guixia, Tang Yun.
ADMET-score – a comprehensive scoring function for evaluation of chemical drug-likeness, MedChemComm, 2019